M1809

MRS 1523

>98% (HPLC)

• Sinonimo/i: 3-Propyl-6-ethyl-5-[(ethylthio)carbonyl]-2 phenyl-4-propyl-3-pyridine carboxylate
• Formula empirica (notazione di Hill): C₂₃H₂₉NO₃S
• Numero CAS: 212329-37-8
• Peso molecolare: 399.55
• NACRES: NA.77
• PubChem Substance ID: 24278127
• UNSPSC Code: 12352200
• MDL number: MFCD03787977
• Assay: >98% (HPLC)
• Form: oil

Proprietà

• Quality Segment: 100
• assay: >98% (HPLC)
• form: oil
• color: colorless to light brown
• solubility: DMSO: >10 mg/mL, H₂O: insoluble
• shipped in: wet ice
• storage temp.: 2-8°C
• SMILES string: CCCOC(=O)c1c(CCC)c(C(=O)SCC)c(CC)nc1-c2ccccc2
• InChI: 1S/C23H29NO3S/c1-5-12-17-19(23(26)28-8-4)18(7-3)24-21(16-13-10-9-11-14-16)20(17)22(25)27-15-6-2/h9-11,13-14H,5-8,12,15H2,1-4H3
• InChI key: UUSHFEVEROROSP-UHFFFAOYSA-N
• Gene Information: human ... ADORA3(140) ; rat ... Adora1(29290), Adora2a(25369), Adora3(25370)

Descrizione

Application

MRS 1523 has been used as an inhibitor of adenosine receptors in SW1990 and BxPC3 pancreatic cancer cells,[1] LX2 human hepatic stellate cells and human coronary smooth muscle cells.[2]

Biochem/physiol Actions

MRS 1523 is a selective adenosine A3 receptor antagonist in the rat.

Features and Benefits

This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Legal Information

Sold under license from the National Institutes of Health

Informazioni sulla sicurezza

• Classe di stoccaggio: 10 - Combustible liquids
• wgk: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable
• ppe: Eyeshields, Gloves