5.08160

DPDPE

• 別名: DPDPE, δ Opioid Receptor Agonist, DPDPE
• 実験式（ヒル表記法）: C₃₀H₃₉N₅O₇S₂
• CAS番号: 88373-73-3
• 分子量: 645.79
• MDL番号: MFCD00076430
• UNSPSCコード: 12352200
• NACRES: NA.77

特性

• アッセイ: ≥99% (HPLC)
• 品質水準: 100
• フォーム: solid
• メーカー／製品名: Calbiochem^®
• 保管条件: OK to freeze; protect from light
• 色: off-white
• 溶解性: water: 1 mg/mL
• 保管温度: −20°C
• SMILES記法: S1SC([C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C1(C)C)C(=O)O)Cc3ccccc3)NC(=O)[C@@H](N)Cc2ccc(cc2)O)(C)C
• InChI: 1S/C30H39N5O7S2/c1-29(2)23(34-25(38)20(31)14-18-10-12-19(36)13-11-18)27(40)32-16-22(37)33-21(15-17-8-6-5-7-9-17)26(39)35-24(28(41)42)30(3,4)44-43-29/h5-13,20-21,23-24,36H,14-16,31H2,1-4H3,(H,32,40)(H,33,37)(H,34,38)(H,35,39)(H,41,42)/t20-,21-,23-,24-/m0/s1
• InChI Key: MCMMCRYPQBNCPH-WMIMKTLMSA-N

詳細

詳細

A potent agonist selective for δ opioid receptor (EC₅₀ = 5.2 nM). Exhibits anti-convulsant effects in vivo in rats, also used in nociceptive studies.

生物化学的／生理学的作用

Primary Target
δ opioid receptor

警告

Toxicity: Standard Handling (A)

シーケンス

Tyr-D-Pen-Gly-Phe-D-Pen (2-5 disulfide bond)

再構成

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.

その他情報

Chen, C., 1997. J. Pharmacol. Exp. Ther.283, 1151.
Chandrakumar, S., et al., 1992. J. Med. Chem.35, 2928.
Tortella, F. 1988. Peptides.9, 1177.
Clark, A., et al., 1986. Eur. J. Pharmacol.128, 303.

法的情報

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

安全性情報

• 保管分類コード: 11 - Combustible Solids
• WGK: WGK 3
• 引火点(°F): Not applicable
• 引火点(℃): Not applicable