推薦產品
化驗
≥97.5% (HPLC)
形狀
powder
顏色
off-white
溶解度
ethanol: ~0.7 mg/mL
DMSO: ~0.9 mg/mL
chloroform: ~10 mg/mL
DMSO: ≤2.6 mg/mL (Achieved with heating.)
ethanol: ≤5 mg/mL (Achieved with heating.)
H2O: insoluble
儲存溫度
room temp
SMILES 字串
O.COc1ccc2C3CC[C@]4(C)[C@H](CCC4C3CCc2c1)NCCCCCCN5C(=O)C=CC5=O
InChI
1S/C29H40N2O3.H2O/c1-29-16-15-23-22-10-8-21(34-2)19-20(22)7-9-24(23)25(29)11-12-26(29)30-17-5-3-4-6-18-31-27(32)13-14-28(31)33;/h8,10,13-14,19,23-26,30H,3-7,9,11-12,15-18H2,1-2H3;1H2/t23-,24-,25+,26+,29+;/m1./s1
InChI 密鑰
WCOYJDRCHHGMRK-BDEPKWELSA-N
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應用
生化／生理作用
抑制 PPI 水解成 IP3，导致细胞溶质游离钙的减少。抑制 G蛋白- 磷脂酶C 活化的偶联，同时保持不受 cAMP 产生的影响。
準備報告
U-73122 水合物可溶于乙醇（约 0.7 mg/ml或 加热时，≤ 5mg/ml）、氯仿（约 10 mg/ml）和DMSO（约 0.9 mg/ml或加热时，≤ 2.6mg/ml）。U-73122 水合物不溶于水。
儲存類別代碼
11 - Combustible Solids
水污染物質分類（WGK）
WGK 3
閃點（°F）
Not applicable
閃點（°C）
Not applicable
個人防護裝備
dust mask type N95 (US), Eyeshields, Gloves
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