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Merck

ADORA2A

adenosine A2a receptor

Sinónimos:
A2aR, ADORA2, RDC8
Especie:
ID UniProtKB:
ID del gen:
  • Human(135) Summary: This gene encodes a member of the guanine nucleotide-binding protein (G protein)-coupled receptor (GPCR) superfamily, which is subdivided into classes and subtypes. The receptors are seven-pass transmembrane proteins that respond to extracellular cues and activate intracellular signal transduction pathways. This protein, an adenosine receptor of A2A subtype, uses adenosine as the preferred endogenous agonist and preferentially interacts with the G(s) and G(olf) family of G proteins to increase intracellular cAMP levels. It plays an important role in many biological functions, such as cardiac rhythm and circulation, cerebral and renal blood flow, immune function, pain regulation, and sleep. It has been implicated in pathophysiological conditions such as inflammatory diseases and neurodegenerative disorders. Alternative splicing results in multiple transcript variants. A read-through transcript composed of the upstream SPECC1L (sperm antigen with calponin homology and coiled-coil domains 1-like) and ADORA2A (adenosine A2a receptor) gene sequence has been identified, but it is thought to be non-coding. [provided by RefSeq, Jun 2013]
  • Mouse(11540) adenosine A2a receptor
  • Rat(25369) adenosine A2a receptor
  • chicken(427705) adenosine A2a receptor
  • naked mole-rat(101718082) adenosine A2a receptor
  • domestic guinea pig(100135473) adenosine A2a receptor
  • sheep(101112926) adenosine A2a receptor
  • cow(617828) adenosine A2a receptor
  • Horse(100034039) adenosine A2a receptor
  • domestic cat(101080742) adenosine A2a receptor
  • dog(403960) adenosine A2a receptor

Custom & Knockdown Gene Products

Small Molecule - Agonist

Número de producto
Descripción
Especie
CGS-21680 hydrochloride hydrate, solid,
Especie
human
Adenosine, ,
Especie
human
Adenosine, United States Pharmacopeia (USP) Reference Standard,
Especie
human
Adenosine, Pharmaceutical Secondary Standard; Certified Reference Material,
Especie
human
Adenosine, phyproof® Reference Substance,
Especie
human

Small Molecule - Antagonist

Número de producto
Descripción
Especie
Istradefylline, ≥98% (HPLC),
Especie
human
3-Isobutil-1-metilxantina, BioUltra, ≥99%,
Especie
rat
Hematoxylin, ,
Especie
rat
Hematoxylin, certified by the BSC,
Especie
rat
3-Methylxanthine, 98%,
Especie
rat

Antibodies

Número de producto
Descripción
Reactividad de especies
Aplicación
Anti-Adenosine Receptor A2a Antibody, clone 7F6-G5-A2, clone 7F6-G5-A2, Upstate®, from mouse,
Reactividad de especies
canine, dog, human, mouse, rabbit, rat
Aplicación
flow cytometry
immunohistochemistry

western blot
Anti-Adenosine A2a Receptor Antibody, Chemicon®, from rabbit,
Reactividad de especies
bovine, canine, human, pig
Aplicación
ELISA
immunocytochemistry

immunohistochemistry

western blot
Anti-Adenosine A2a Receptor Antibody, serum, Chemicon®,
Reactividad de especies
bovine, canine, human, pig, rat
Aplicación
ELISA
western blot
Anti-ADORA2A (C-terminal) antibody produced in rabbit, affinity isolated antibody,
Reactividad de especies
bovine, canine, guinea pig, horse, human, mouse, rabbit, rat
Aplicación
immunohistochemistry
western blot
Anti-AA2AR / Adenosine A2aR Reference Antibody, ,
Reactividad de especies
human
Aplicación

Small Molecule - Inhibitor

Número de producto
Descripción
Especie
EHNA hydrochloride, ≥98% (HPLC),
Especie
human
Dilazep dihydrochloride, powder,
Especie
human
8-(3-Chlorostyryl)caffeine, ≥98% (HPLC), solid,
Especie
human, rat, mouse
5′-Deoxy-5′-(methylthio)adenosine, ,
Especie
human, rat, mouse
α-Naphthoflavone, ≥98%,
Especie
human, rat

Small Molecule - Ligand

Número de producto
Descripción
Especie
2-Chloro-2′-deoxyadenosine, antileukemic,
Especie
rat, human
1,7-Dimethylxanthine, ~98%, solid,
Especie
rat, human
Chloro-IB-MECA, solid, ≥98% (HPLC),
Especie
human, rat
Adenosine, ≥99%,
Especie
human, rat
Theophylline, anhydrous, ≥99%, powder,
Especie
mouse, human, rat

Small Molecule - Mixed Agonist/Antagonist

Número de producto
Descripción
Especie
2-Iodoadenosine, 97%,
Especie
human, rat
2-Fluoroadenine-9-β-D-arabinofuranoside, DNA synthesis and methylation inhibitor,
Especie
rat, human
2-Fluoroadenosine, 97%,
Especie
rat, human
2-Chloroadenosine, ,
Especie
human, rat
Chloro-IB-MECA, solid, ≥98% (HPLC),
Especie
human, rat

esiRNA

Número de producto
Descripción
Especie
MISSION® esiRNA, targeting human ADORA2A, SPECC1L-ADORA2A,
Especie
human
MISSION® esiRNA, targeting mouse Adora2a,
Especie
mouse