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Merck
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文件

A0862

Sigma-Aldrich

A-740003

≥98% (HPLC)

同義詞:

N-(1-{[(氰亚胺基)(5-喹啉氨基)甲基] 氨基 }-2,2-二甲基丙基)-2-(3,4-二甲氧基苯基)乙酰胺

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About This Item

經驗公式(希爾表示法):
C26H30N6O3
CAS號碼:
分子量::
474.55
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77

品質等級

化驗

≥98% (HPLC)

形狀

powder

顏色

white to light brown

溶解度

DMSO: 10 mg/mL, clear (warmed)

儲存溫度

2-8°C

SMILES 字串

COc1ccc(CC(=O)NC(N\C(Nc2cccc3ncccc23)=N\C#N)C(C)(C)C)cc1OC

InChI

1S/C26H30N6O3/c1-26(2,3)24(31-23(33)15-17-11-12-21(34-4)22(14-17)35-5)32-25(29-16-27)30-20-10-6-9-19-18(20)8-7-13-28-19/h6-14,24H,15H2,1-5H3,(H,31,33)(H2,29,30,32)

InChI 密鑰

PUHSRMSFDASMAE-UHFFFAOYSA-N

一般說明

A-740003 是一种高度仿射和选择性 P2X7 受体拮抗剂,最适合于放射性示踪剂进展,用于正电子发射断层扫描神经炎症成像。

生化/生理作用

A-740003 是一种选择性 P2X7 嘌呤受体拮抗剂。

特點和優勢

该化合物的相关信息整理于受体分类和信号转导手册的 P2受体:P2X离子通道家族 页面。欲浏览其他手册页面,请 点击这里

儲存類別代碼

11 - Combustible Solids

水污染物質分類(WGK)

WGK 3

閃點(°F)

Not applicable

閃點(°C)

Not applicable


分析證明 (COA)

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