Accéder au contenu
Merck

ABCB1

ATP-binding cassette, sub-family B (MDR/TAP), member 1

Synonymes:
ABC20, CD243, CLCS, GP170, MDR1, P-GP, PGY1
Espèce(s):
ID UniProtKB:
ID du gène:
  • Human(5243) Summary: The membrane-associated protein encoded by this gene is a member of the superfamily of ATP-binding cassette (ABC) transporters. ABC proteins transport various molecules across extra- and intra-cellular membranes. ABC genes are divided into seven distinct subfamilies (ABC1, MDR/TAP, MRP, ALD, OABP, GCN20, White). This protein is a member of the MDR/TAP subfamily. Members of the MDR/TAP subfamily are involved in multidrug resistance. The protein encoded by this gene is an ATP-dependent drug efflux pump for xenobiotic compounds with broad substrate specificity. It is responsible for decreased drug accumulation in multidrug-resistant cells and often mediates the development of resistance to anticancer drugs. This protein also functions as a transporter in the blood-brain barrier. [provided by RefSeq, Jul 2008]
  • dog(403879) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • domestic cat(493707) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • Thale Cress(818265) ABC transporter B family member 1
  • naked mole-rat(101702843) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • domestic guinea pig(100733532) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • Domestic Rabbit(100008914) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • sheep(443367) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • Horse(100034074) ATP-binding cassette, sub-family B (MDR/TAP), member 1
  • cow(281585) ATP-binding cassette, sub-family B (MDR/TAP), member 1

Custom & Knockdown Gene Products

  • siRNA

    Shop predesigned siRNA that are designed using the proprietary Rosetta Inpharmatics algorithm.

  • shRNA

    Shop the largest, most validated shRNA collection and build your own clone sets.

  • Custom Gene Products

    We offer a comprehensive portfolio of DNA oligos, RNA oligos and predesigned primers.

Small Molecule - Agonist

Référence du produit
Description
Espèce(s)
9(10H)-Acridanone, 99%,
Espèce(s)
human
Hydrocortisone, BioReagent, suitable for cell culture,
Espèce(s)
human, mouse, rat
Hydrocortisone solution, 50 μM, sterile-filtered, BioXtra, suitable for cell culture,
Espèce(s)
human, mouse, rat
Hydrocortisone, γ-irradiated, powder, BioXtra, suitable for cell culture,
Espèce(s)
human, mouse, rat
Hydrocortisone, ≥98% (HPLC),
Espèce(s)
human, mouse, rat

Small Molecule - Antagonist

Référence du produit
Description
Espèce(s)
Chlorosulfonyl isocyanate, 98%,
Espèce(s)
human
Omeprazole, solid,
Espèce(s)
human
Erythromycin, BioReagent, suitable for cell culture,
Espèce(s)
mouse, human
Clotrimazole, ,
Espèce(s)
mouse, human
Erythromycin, potency: ≥850 μg per mg,
Espèce(s)
mouse, human

Antibodies

Référence du produit
Description
Espèces réactives
Application
Monoclonal Anti-P-Glycoprotein (MDR) antibody produced in mouse, clone F4, ascites fluid,
Espèces réactives
hamster, human
Application
ELISA
immunocytochemistry

immunohistochemistry

immunoprecipitation (IP)

radioimmunoassay

western blot
Anti-MDR-1 Antibody, clone 1O12 ZooMAb® Rabbit Monoclonal, recombinant, expressed in HEK 293 cells,
Espèces réactives
human, mouse
Application
affinity binding assay
flow cytometry

immunocytochemistry

immunohistochemistry

western blot
Anti-ABCB1 antibody produced in rabbit, Prestige Antibodies® Powered by Atlas Antibodies, affinity isolated antibody, buffered aqueous glycerol solution,
Espèces réactives
human
Application
immunofluorescence
immunohistochemistry
Anti-MDR1 Antibody, clone JSB-1, culture supernatant, clone JSB-1, Chemicon®,
Espèces réactives
hamster, human
Application
flow cytometry
immunocytochemistry

immunohistochemistry

western blot
Anti-MDR1 Antibody, extracellular human specific Pgp, clone MC57, clone MC57, Chemicon®, from mouse,
Espèces réactives
human
Application
flow cytometry
immunohistochemistry

Cell Lines

Référence du produit
Description
Espèce(s)
CAR Knockout HepaRG Cells, 1 vial,
Espèce(s)
MDR1 Knockout Caco-2 Cells, one vial,
Espèce(s)
human
MDR1 Knockout HepaRG Cells, 1 vial,
Espèce(s)
human
MDR1/MRP2 Double Knockout Caco-2 Cells, one vial,
Espèce(s)
human

Kits

Référence du produit
Description
Espèce(s)
Multidrug Resistance Assay Kit, (Fluorometric MDR Assay),
Espèce(s)
human, mouse, rat

Small Molecule - Mixed Agonist/Antagonist

Référence du produit
Description
Espèce(s)
Dexaméthasone, powder, BioReagent, suitable for cell culture, ≥97%,
Espèce(s)
mouse, rat, human
Dexaméthasone, ≥98% (HPLC), powder,
Espèce(s)
mouse, rat, human
Dexaméthasone, powder, γ-irradiated, BioXtra, suitable for cell culture, ≥80% (HPLC),
Espèce(s)
mouse, rat, human
Progesterone-Water Soluble, powder, BioReagent, suitable for cell culture,
Espèce(s)
mouse, human, rat
Dexaméthasone, meets USP testing specifications,
Espèce(s)
mouse, rat, human

Proteins

Référence du produit
Description
Espèce(s)
SB-MDR1-Hi5-PREDEASY-ATPase kit, membrane based kit for Human MDR1 ATPase Transport Assays,
Espèce(s)
human

esiRNA

Référence du produit
Description
Espèce(s)
MISSION® esiRNA, targeting human ABCB1,
Espèce(s)
human