SML0342

TFM-4AS-1

≥98% (HPLC)

• Synonym(e): (4aR,6aS,7S,11aR)-1,4a,6a-Trimethyl-2-oxo-N-[2-(trifluoromethyl)phenyl]-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11atetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxamide
• Empirische Formel (Hill-System): C₂₇H₃₃F₃N₂O₂
• CAS-Nummer: 188589-61-9
• Molekulargewicht: 474.56
• UNSPSC Code: 51111800
• PubChem Substance ID: 329825347
• NACRES: NA.77
• Assay: ≥98% (HPLC)
• Form: powder
• Quality level: 100

Eigenschaften

• SMILES string: CN1[C@@H]2CC[C@@H]3[C@@H]4CC[C@H](C(=O)Nc5ccccc5C(F)(F)F)[C@@]4(C)CC[C@@H]3[C@@]2(C)C=CC1=O
• InChI: 1S/C27H33F3N2O2/c1-25-14-12-18-16(8-11-22-26(18,2)15-13-23(33)32(22)3)17(25)9-10-20(25)24(34)31-21-7-5-4-6-19(21)27(28,29)30/h4-7,13,15-18,20,22H,8-12,14H2,1-3H3,(H,31,34)/t16-,17+,18+,20-,22-,25+,26-/m1/s1
• InChI key: YFBLEKKYWFJKBP-HNXMFXTHSA-N
• assay: ≥98% (HPLC)
• form: powder
• color: white to beige
• solubility: DMSO: >5 mg/mL
• storage temp.: 2-8°C
• Quality Level: 100

Beschreibung

Biochem/physiol Actions

TFM-4AS-1 is a potent SARM (Selective Androgen Receptor Modulator) and partial agonist of AR.

TFM-4AS-1 is a potent SARM (Selective Androgen Receptor Modulator). TFM-4AS-1 is a partial agonist of AR. The compound promotes the buildup of bone and muscle mass while having reduced effects on reproductive organs and sebaceous glands. The compound also is an inhibitor of rat 5 α-reductase enzymes type I (2 nM) and type 2 (3 nM).

Sicherheitshinweise

• Lagerklasse: 11 - Combustible Solids
• wgk: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable