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About This Item
經驗公式(希爾表示法):
C20H20N2O2
CAS號碼:
分子量::
320.39
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77
暫時無法取得訂價和供貨情況
推薦產品
品質等級
化驗
≥98% (HPLC)
形狀
powder
顏色
white to beige
溶解度
DMSO: 5 mg/mL, clear (warmed)
儲存溫度
2-8°C
SMILES 字串
CC1=NC2=C(NC(C3=CC=C(OC(C)C)C=C3)=O)C=CC=C2C=C1
InChI
1S/C20H20N2O2/c1-13(2)24-17-11-9-16(10-12-17)20(23)22-18-6-4-5-15-8-7-14(3)21-19(15)18/h4-13H,1-3H3,(H,22,23)
InChI 密鑰
GVGVYDCVFBGALZ-UHFFFAOYSA-N
生化/生理作用
CDN1163处理可降低与糖异生和脂肪生成有关的基因的肝表达,同时减弱内质网(ER)应激反应和ER应激诱导的细胞凋亡。[1]CDN1163可与肌膜/内质网Ca2+-ATPase(SERCA)发生相互作用,并增强ER Ca2+的内含量。[2]
CDN1163是肌/内质网Ca2+-ATPase(SERCA)的一种变构激活剂。
CDN1163是肌/内质网Ca2+-ATPase(SERCA)的一种变构激活剂,可有效降低ob/ob小鼠的空腹血糖,改善的葡萄糖耐量和肝脂肪变性。另外,CDN1163可诱导肥胖组织重量显著减少,而对ob/ob小鼠的瘦体重没有影响。CDN1163对瘦对照小鼠的葡萄糖水平或体重没有影响。
儲存類別代碼
11 - Combustible Solids
水污染物質分類(WGK)
WGK 3
閃點(°F)
Not applicable
閃點(°C)
Not applicable
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分析證明 (COA)
Lot/Batch Number
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