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Merck

A6226

Sigma-Aldrich

AM251

>98% (HPLC), solid, cannabinoid receptor (CB1) antagonist

别名:

1-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-1-哌啶基-1H-吡唑-3-甲酰胺

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About This Item

经验公式(希尔记法):
C22H21N4OCl2I
分子量:
555.24
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77

product name

AM251, >98% (HPLC), solid

品質等級

化驗

>98% (HPLC)

形狀

solid

顏色

white

溶解度

DMSO: >10 mg/mL
H2O: insoluble

起源

Sanofi Aventis

SMILES 字串

Cc1c(nn(-c2ccc(Cl)cc2Cl)c1-c3ccc(I)cc3)C(=O)NN4CCCCC4

InChI

1S/C22H21Cl2IN4O/c1-14-20(22(30)27-28-11-3-2-4-12-28)26-29(19-10-7-16(23)13-18(19)24)21(14)15-5-8-17(25)9-6-15/h5-10,13H,2-4,11-12H2,1H3,(H,27,30)

InChI 密鑰

BUZAJRPLUGXRAB-UHFFFAOYSA-N

基因資訊

應用

AM251,一种CB1 大麻素受体拮抗剂,已被用于一项研究,以确定其与海马神经元的相互作用,以增强小鼠的空间记忆。

生化/生理作用

AM251是一种CB1 大麻素受体拮抗剂。

特點和優勢

《受体分类和信号转导》手册的大麻素受体页有该化合物的介绍。想要浏览手册的其他页面, 请单击此处
该化合物由Sanofi Aventis开发。要浏览其他药物开发化合物和批准的药物/候选药物列表,单击此处

其他說明

盐含量可能会有所不同。

危險聲明

防範說明

危險分類

Aquatic Chronic 4

儲存類別代碼

11 - Combustible Solids

水污染物質分類(WGK)

WGK 3

閃點(°F)

Not applicable

閃點(°C)

Not applicable

個人防護裝備

dust mask type N95 (US), Eyeshields, Gloves


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