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Merck
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文件

371725

Sigma-Aldrich

GPR43（FFA2）激动剂

The GPR43 (FFA2) Agonist controls the biological activity of GPR43. This small molecule/inhibitor is primarily used for Biochemicals applications.

别名:

GPR43（FFA2）激动剂, （S）-2-（4-氯苯基）-3，3-二甲基-N-（5-苯基噻唑-2-基）丁酰胺

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About This Item

经验公式（希尔记法）:
C21H21ClN2OS
CAS号:
1208552-99-1
分子量:
384.92
分類程式碼代碼:
51111800
NACRES:
NA.77

品質等級

100

化驗

>98% (HPLC)

形狀

solid

製造商／商標名

Calbiochem®

儲存條件

OK to freeze

顏色

white

溶解度

DMSO: 50 mg/mL

運輸包裝

ambient

儲存溫度

2-8°C

一般說明

一种苯乙酰胺化合物，可作为FFA2的变构激动剂（GPR43），在hFFA2毛喉素诱导的cAMP分析中显示出相对于乙酸盐的左移乙酸盐剂量反应（IC50 = 0.7 µM）和111%的功效。

警告

毒性：标准处理（A）

重構

复溶后，等分并冷冻保存（-20°C）。储备溶液在-20°C下可稳定保存至多3个月。

其他說明

Wang, Y., et al. 2009.Bioorg.Med. Chem. Lett.20, 493.

法律資訊

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

儲存類別代碼

11 - Combustible Solids

水污染物質分類（WGK）

WGK 3

閃點（°F）

Not applicable

閃點（°C）

Not applicable

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