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SML0790

Iperoxo

Name: Iperoxo
Brand: SIGMA

≥98% (HPLC), Acetylcholine receptor agonist, powder

Synonym(e):

4-[(4,5-Dihydro-3-isoxazolyl)oxy]-N,N,N-trimethyl-2-butyn-1-aminium iodide

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Über diesen Artikel

Empirische Formel (Hill-System):

C₁₀H₁₇IN₂O₂

CAS-Nummer:

247079-84-1

Molekulargewicht:

324.16

UNSPSC Code:

12352200

NACRES:

NA.77

Assay:

≥98% (HPLC)

Form:

powder

Technischer Dienst

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Eigenschaften

Produktname

Iperoxo, ≥98% (HPLC)

Quality Segment

100

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

H₂O: 5 mg/mL, clear (warmed)

storage temp.

2-8°C

InChI

1S/C9H14N2O2/c1-11(2)6-3-4-7-12-9-5-8-13-10-9/h5-8H2,1-2H3

InChI key

CADHNBBPGYVTOA-UHFFFAOYSA-N

Beschreibung

Biochem/physiol Actions

Iperoxo is a muscarinic acetylcholine receptor superagonist.

Iperoxo is a muscarinic acetylcholine receptor superagonist. The pEC₅₀ values for G-protein activation by acetylcholine and iperoxo in CHO cells expressing recombinant human M2 receptors are 7.6 and 10.1, respectively.

Iperoxo forms an important building block for the class of G protein-coupled receptors modulators. Iperoxo specifically binds to the orthosteric site of the muscarinic acetylcholine receptor. It has a higher efficacy than the endogenous agonist acetylcholine.

Features and Benefits

This compound is a featured product for Neuroscience research. Click here to discover more featured Neuroscience products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

This compound is featured on the Acetylcholine Receptors (Muscarinic) page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.