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PZ0229

Sigma-Aldrich

PF-03246799 hydrochloride

≥98% (HPLC)

Synonym(s):

6,7,8,9-Tetrahydro-2-(phenylmethyl)-5H-pyrimido[4,5-d]azepine hydrochloride, PF-3246799 hydrochloride

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5 MG
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25 MG
$291.00

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5 MG
$103.00
25 MG
$291.00

About This Item

Empirical Formula (Hill Notation):
C15H17N3 · xHCl
CAS Number:
Molecular Weight:
239.32 (free base basis)
UNSPSC Code:
51111800
PubChem Substance ID:
NACRES:
NA.77

$103.00


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Quality Level

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

H2O: 20 mg/mL, clear

storage temp.

room temp

SMILES string

C1(CC2=NC(CCNCC3)=C3C=N2)=CC=CC=C1.Cl

InChI

1S/C15H17N3.ClH/c1-2-4-12(5-3-1)10-15-17-11-13-6-8-16-9-7-14(13)18-15;/h1-5,11,16H,6-10H2;1H

InChI key

ICVPRIZGSIUCOE-UHFFFAOYSA-N

Biochem/physiol Actions

PF-3246799 is a potent serotonin 5-HT2C receptor agonist with an EC50 of 4.5 nM and minimal activity at 5-HT2A and 5-HT2B receptors. PF-3246799 had good efficacy in a preclinical canine model of stress urinary incontinence.
PF-3246799 is a potent serotonin 5-HT2C receptor agonist.

Features and Benefits

This compound is a featured product for Neuroscience research. Click here to discover more featured Neuroscience products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

Storage Class

11 - Combustible Solids

wgk_germany

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable


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