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SML3334

Ceefourin 1

≥95% (HPLC)

Synonym(s):

5-[(2-Benzothiazolylthio)methyl]-2,4-dihydro-4-methyl-3H-1,2,4-triazole-3-thione, Ceefourin-1

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About This Item

Empirical Formula (Hill Notation):
C11H10N4S3
CAS Number:
315702-40-0
Molecular Weight:
294.42
UNSPSC Code:
12352200
NACRES:
NA.77
MDL number:
MFCD02329957
Assay:
≥95% (HPLC)
Form:
powder
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Quality Segment

100

assay

≥95% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 2 mg/mL, clear

storage temp.

-10 to -25°C

SMILES string

CN1C(CSC2=NC3=C(C=CC=C3)S2)=NNC1=S

Biochem/physiol Actions

Ceefourin 1 is a potent and highly selective MRP4 (Multidrug resistance protein 4) inhibitor that exhibits low cellular toxicity and high microsomal and acid stability. Ceefourin 1 inhibits PDAC (pancreatic ductal adenocarcinoma) cell proliferation through MRP4-dependent cAMP extrusion thereby activation of the cAMP/Epac/Rap1 signaling pathway.
Potent and highly selective MRP4 (Multidrug resistance protein 4) inhibitor

Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

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