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Key Documents

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C102

Sigma-Aldrich

8-Cyclopentyl-1,3-dimethylxanthine

≥98% (HPLC), powder

Sinónimos:

8-Cyclopentyltheophylline, CPT

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About This Item

Fórmula empírica (notación de Hill):
C12H16N4O2
Número de CAS:
35873-49-5
Peso molecular:
248.28
MDL number:
MFCD00055116
UNSPSC Code:
12352200
PubChem Substance ID:
24277730
NACRES:
NA.77

assay

≥98% (HPLC)

form

powder

color

white to off-white

solubility

H2O: slightly soluble <0.28 mg/mL
45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.77 mg/mL
DMSO: ~16 mg/mL at 60 °C
0.1 M NaOH: soluble

SMILES string

CN1C(=O)N(C)c2nc([nH]c2C1=O)C3CCCC3

InChI

1S/C12H16N4O2/c1-15-10-8(11(17)16(2)12(15)18)13-9(14-10)7-5-3-4-6-7/h7H,3-6H2,1-2H3,(H,13,14)

InChI key

SCVHFRLUNIOSGI-UHFFFAOYSA-N

Gene Information

human ... ADORA1(134)

Biochem/physiol Actions

Selective A1 adenosine receptor antagonist.

Features and Benefits

This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Storage Class

11 - Combustible Solids

wgk_germany

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

Certificados de análisis (COA)

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