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Merck

G5918

Sigma-Aldrich

GR 113808

≥98% (HPLC), solid

别名:

1-[2-[(甲磺酰基)氨基]乙基]-4-哌啶基]甲基1-甲基-1H-吲哚-3-羧酸酯

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About This Item

经验公式(希尔记法):
C19H27N3O4S
分子量:
393.50
MDL號碼:
分類程式碼代碼:
12352200
PubChem物質ID:
NACRES:
NA.77

化驗

≥98% (HPLC)

形狀

solid

顏色

white to light pink

溶解度

DMSO: >20 mg/mL

起源

GlaxoSmithKline

儲存溫度

2-8°C

SMILES 字串

Cn1cc(C(=O)OCC2CCN(CCNS(C)(=O)=O)CC2)c3ccccc13

InChI

1S/C19H27N3O4S/c1-21-13-17(16-5-3-4-6-18(16)21)19(23)26-14-15-7-10-22(11-8-15)12-9-20-27(2,24)25/h3-6,13,15,20H,7-12,14H2,1-2H3

InChI 密鑰

MOZPSIXKYJUTKI-UHFFFAOYSA-N

基因資訊

應用

GR 113808已被用作5-羟色胺受体4(5-HT4R)阻断剂,以研究其对大鼠心室心肌细胞中钙(Ca2+)瞬变的影响。它也已被用作5-HT4R拮抗剂,以研究其对胚胎后斑马鱼从头肠神经发生的影响。

生化/生理作用

GR 113808是5-HT4血清素受体拮抗剂。

特點和優勢

该化合物由 GlaxoSmithKline开发。想浏览其他制药公司开发的化合物和已批准药物/候选药物目录, 请单击此处

法律資訊

根据Glaxo­Smith­Kline的协议出售用于研究目的

儲存類別代碼

11 - Combustible Solids

水污染物質分類(WGK)

WGK 3

閃點(°F)

Not applicable

閃點(°C)

Not applicable

個人防護裝備

Eyeshields, Gloves, type N95 (US)


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