R134

Rilmenidine hemifumarate salt

solid

• Synonym(s): N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt, Oxaminozoline hemifumarate salt, Rilmenidene hemifumarate salt
• Empirical Formula (Hill Notation): C₁₀H₁₆N₂O · 0.5C₄H₄O₄
• CAS Number: 207572-68-7
• Molecular Weight: 238.28
• NACRES: NA.77
• PubChem Substance ID: 24277752
• UNSPSC Code: 12352200
• MDL number: MFCD09878261
• Form: solid

Properties

• form: solid
• Quality Segment: 100
• color: white
• solubility: DMSO: >10 mg/mL, H₂O: insoluble
• originator: Servier
• SMILES string: OC(=O)\C=C\C(O)=O.C1CN=C(NC(C2CC2)C3CC3)O1.C4CN=C(NC(C5CC5)C6CC6)O4
• InChI: 1S/2C10H16N2O.C4H4O4/c2*1-2-7(1)9(8-3-4-8)12-10-11-5-6-13-10;5-3(6)1-2-4(7)8/h2*7-9H,1-6H2,(H,11,12);1-2H,(H,5,6)(H,7,8)/b;;2-1+
• InChI key: LZFATBMLSYHRTC-WXXKFALUSA-N
• Gene Information: human ... NISCH(11188)

Description

Biochem/physiol Actions

Selective I₁ imidazoline receptor agonist.

Features and Benefits

This compound is featured on the Imidazoline Binding Sites page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

This compound was developed by Servier. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Safety Information

• wgk: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable
• ppe: Eyeshields, Gloves, type N95 (US)
• pictograms: GHS06
• signalword: Danger
• hcodes: H301
• pcodes: P264 - P270 - P301 + P310 - P405 - P501
• Hazard Classifications: Acute Tox. 3 Oral
• Storage Class: 6.1C - Combustible acute toxic Cat.3 / toxic compounds or compounds which causing chronic effects