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Key Documents

657021

Sigma-Aldrich

Tyrosine Kinase Inhibitor Set II

The Tyrosine Kinase Inhibitor Set II controls the biological activity of Tyrosine Kinase. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

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About This Item

UNSPSC 코드:
12352200

Quality Level

형태

solid

제조업체/상표

Calbiochem®

저장 조건

OK to freeze
protect from light

배송 상태

ambient

저장 온도

−20°C

일반 설명

Contains 20 mg of Genistein (Cat. No. 345834), 1 mg of PP2 (Cat. No. 529573), 5 mg of AG 490 (Cat. No. 658401), 5 mg of AG 1296 (Cat. No. 658551), and 5 mg of AG 1478 (Cat. No. 658552). Supplied with an informational insert.
Protein tyrosine phosphorylation is a key element in several membrane signal transduction systems. There are two general classes of tyrosine kinases: the receptor tyrosine kinases and the receptor-associated tyrosine kinases. The receptor tyrosine kinases possess an extracellular ligand binding domain and an intracellular catalytic domain with intrinsic tyrosine kinase activity. The receptor-associated tyrosine kinases transmit signals from the membrane by interacting with the cytoplasmic domain of membrane proteins.



The design of specific inhibitors of tyrosine kinases is important for both fundamental research and for developing therapeutic strategies for the treatment of cancer, atherosclerosis, psoriasis, septic shock, and other disorders where increased tyrosine kinase activity has been reported.



The Tyrosine Kinase Inhibitor Set contains a general tyrosine kinase inhibitor and a series of other inhibitors, which are selective for various tyrosine kinases that are important in cellular signaling. The set contents and characteristics are listed in the table below.

생화학적/생리학적 작용

Product competes with ATP.
Secondary Target
PKC, Src family of protein tyrosine kinases, JAK2

포장

Packaged under inert gas

경고

Toxicity: Standard Handling (A)

제조 메모

Concentrated solutions of ≥1 mg/ml should be prepared in anhydrous DMSO.

기타 정보

Hanke, J.H., et al. 1996. J. Biol. Chem.271 695.
Meydan, N., et al. 1996. Nature379, 645.
Levitzi, A., and Gazit, A. 1995. Science267, 1782.
Akiyama, T., et al. 1987. J. Biol. Chem.262, 5592.

법적 정보

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

픽토그램

Exclamation mark

신호어

Warning

유해 및 위험 성명서

예방조치 성명서

Hazard Classifications

Acute Tox. 4 Oral

Storage Class Code

11 - Combustible Solids


시험 성적서(COA)

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