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Copper-mediated N-cyclopropylation of azoles, amides, and sulfonamides by cyclopropylboronic acid.

The Journal of organic chemistry (2008-07-10)
Sébastien Bénard, Luc Neuville, Jieping Zhu
ABSTRACT

Reaction of azoles, amides, and sulfonamides in dichloroethane with readily available cyclopropylboronic acid in the presence of copper acetate and sodium carbonate afforded the N-cyclopropyl derivatives in good to excellent yields.

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Sigma-Aldrich
Cyclopropylboronic acid