Design and synthesis of potent N1-substituted indole melatonin receptor agonists.

Design and synthesis of potent N1-substituted indole melatonin receptor agonists.

Chemical communications (Cambridge, England) (2003-03-05)

Andrew Tsotinis, Andreas Eleutheriades, Katherine Hough, David Sugden

摘要

The design and expeditious synthesis of two new indole analogs with up to 5-fold potency of that of melatonin is described.