Z0878
Zaprinast
cGMP-specific phosphodiesterases V and VI inhibitor, solid
Synonym(s):
1,4-Dihydro-5-(2-propoxyphenyl)-7H-1,2,3-triazolo(4,5-d)pyrimidin-7-one
Select a Size
| Size/SKU | Availability | Price |
|---|---|---|
25 mg | Please contact Customer Service for Availability | CZK 2,550.00 |
100 mg | Please contact Customer Service for Availability | CZK 8,590.00 CZK 7,301.50 |
About This Item
CZK 2,550.00
Product Name
Zaprinast, solid
form
solid
Quality Segment
color
white
solubility
45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.11 mg/mL, DMSO: 10 mg/mL, H2O: insoluble
SMILES string
CCCOc1ccccc1C2=NC(=O)c3nn[nH]c3N2
InChI
1S/C13H13N5O2/c1-2-7-20-9-6-4-3-5-8(9)11-14-12-10(13(19)15-11)16-18-17-12/h3-6H,2,7H2,1H3,(H2,14,15,16,17,18,19)
InChI key
REZGGXNDEMKIQB-UHFFFAOYSA-N
Gene Information
human ... PDE2A(5138), PDE4A(5141), PDE4B(5142), PDE4D(5144)
Application
Biochem/physiol Actions
1 of 1
This Item | |||
|---|---|---|---|
| form solid | form powder | form solid | form powder |
| Quality Level 200 | Quality Level 200 | Quality Level 100 | Quality Level 200 |
| solubility 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 0.11 mg/mL, H2O: insoluble, DMSO: 10 mg/mL | solubility 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: soluble 23.3 mg/mL, methanol: soluble 25 mg/mL, clear, colorless, 0.1 M HCl: soluble 7.4 mg/mL, DMSO: soluble, H2O: soluble, hazy, colorless | solubility DMSO: 2 mg/mL, 2-hydroxypropyl-β-cyclodextrin: insoluble, H2O: insoluble, ethanol: insoluble | solubility methanol: 62.5 mg/mL, 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: insoluble, H2O: insoluble |
| color white | color - | color white | color off-white to yellow |
| Gene Information human ... PDE2A(5138), PDE4A(5141), PDE4B(5142), PDE4D(5144) | Gene Information human ... HTR1A(3350), HTR1B(3351), HTR1D(3352), HTR1E(3354), HTR1F(3355), HTR2A(3356), HTR2C(3358), SLC6A4(6532) | Gene Information human ... ADORA3(140) | Gene Information human ... ADORA3(140), CACNA1C(775), CACNA1D(776), CACNA1F(778), CACNA1S(779), CACNG1(786), NR3C2(4306) |
signalword
Warning
hcodes
Hazard Classifications
Eye Irrit. 2 - Skin Irrit. 2 - STOT SE 3
target_organs
Respiratory system
Storage Class
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
ppe
dust mask type N95 (US), Eyeshields, Gloves
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