Skip to Content
Merck

Skip To

SML1784

BTI-A-404

≥98% (HPLC)

Synonym(s):

4-[4-(Dimethylamino)phenyl]-N-(3,5-dimethylphenyl)-1,2,3,4-tetrahydro-6-methyl-2-oxo-5-pyrimidinecarboxamide

Sign In to View Organizational & Contract Pricing.

Select a Size

Change View
Size/SKUAvailabilityPrice
5 mg
Please contact Customer Service for Availability
2 430,00 CZK
2 065,50 CZK

About This Item

Empirical Formula (Hill Notation):
C22H26N4O2
CAS Number:
Molecular Weight:
378.47
UNSPSC Code:
51111800
PubChem Substance ID:
NACRES:
NA.77
Assay:
≥98% (HPLC)
Form:
powder

2 065,50 CZK

List Price2 430,00 CZKSave 15%
Web-Only Promotion

Please contact Customer Service for Availability

​
Technical Service
Need help? Our team of experienced scientists is here for you.
Let Us Assist


Quality Segment

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 5 mg/mL, clear (warmed)

storage temp.

2-8°C

SMILES string

O=C1NC(C2=CC=C(N(C)C)C=C2)C(C(NC3=CC(C)=CC(C)=C3)=O)=C(C)N1

InChI key

JQVNMIXFWKEYQJ-UHFFFAOYSA-N

Biochem/physiol Actions

BTI-A-404 is a potent and selective competitive inverse agonist of human GPR43 (FFAR2).
BTI-A-404 is a potent and selective competitive inverse agonist of human GPR43 (GPR43/Free Fatty Acid Receptor 2, FFAR2) that increases the cyclic AMP level and regulates and reduces acetate-induced cytoplasmic Ca2+ level. BTI-A-404 regulates the downstream signaling pathways of GPR43, including ERK, p38 MAPK, and NF-KB. BTI-A-404 stimulates GLP-1 release.

Compare Similar Items

View Full Comparison

Show Differences

1 of 1

This Item
371725ABC299SAB2109184
description

≥98% (HPLC)

description

The GPR43 (FFA2) Agonist controls the biological activity of GPR43. This small molecule/inhibitor is primarily used for Biochemicals applications.

description

from rabbit, purified by affinity chromatography

description

affinity isolated antibody

assay

≥98% (HPLC)

assay

>98% (HPLC)

assay

-

assay

-

form

powder

form

solid

form

-

form

buffered aqueous solution

Quality Level

100

Quality Level

100

Quality Level

100

Quality Level

-

storage temp.

2-8°C

storage temp.

2-8°C

storage temp.

-

storage temp.

−20°C

solubility

DMSO: 5 mg/mL, clear (warmed)

solubility

DMSO: 50 mg/mL

solubility

-

solubility

-

color

white to beige

color

white

color

-

color

-


Storage Class

11 - Combustible Solids

WGK

WGK 3

Flash Point (°F)

Not applicable

Flash Point (°C)

Not applicable



Choose from one of the most recent versions:

Certificates of Analysis (COA)

Lot/Batch Number

It looks like we've run into a problem, but you can still download Certificates of Analysis from our Documents section.

If you need assistance, please contact Customer Support

Already Own This Product?

Find documentation for the products that you have recently purchased in the Document Library.

Visit the Document Library




Questions

Reviews

No rating value

Active Filters