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E3263

Efaroxan hydrochloride

≥98% (HPLC)

Synonym(s):

2-Ethyl-2-(imidazolin-2-yl)-2,3-dihydrobenzofuran hydrochloride, RX 821037A

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Size/SKUAvailabilityPrice
10 mg
Please contact Customer Service for Availability
CZK 2,710.00
CZK 2,303.50
50 mg
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CZK 8,680.00
CZK 7,378.00

About This Item

Empirical Formula (Hill Notation):
C13H16N2O · HCl
CAS Number:
89197-00-2
Molecular Weight:
252.74
NACRES:
NA.77
PubChem Substance ID:
24278415
UNSPSC Code:
12352200
MDL number:
MFCD00069270
Assay:
≥98% (HPLC)

CZK 2,303.50

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Quality Segment

100

assay

≥98% (HPLC)

solubility

H2O: >20 mg/mL

SMILES string

Cl.CCC1(Cc2ccccc2O1)C3=NCCN3

InChI

1S/C13H16N2O.ClH/c1-2-13(12-14-7-8-15-12)9-10-5-3-4-6-11(10)16-13;/h3-6H,2,7-9H2,1H3,(H,14,15);1H

InChI key

DWOIUCRHVWIHAH-UHFFFAOYSA-N

Gene Information

human ... ADRA1A(148), ADRA1B(147), ADRA1D(146), ADRA2A(150), ADRA2B(151), ADRA2C(152)

Biochem/physiol Actions

(+)-Isomer is a selective α-adrenoceptor antagonist; (−)-isomer is an imidazoline ligand that induces insulin secretion, mediated by the blockade of ATP-sensitive potassium channels in pancreatic β cells; I1 imidazoline binding site antagonist.
(+)-Isomer is a selective α-adrenoceptor antagonist; (−)-isomer is an imidazoline ligand; I1 imidazoline binding site antagonist.

Features and Benefits

This compound is featured on the Imidazoline Binding Sites and Potassium Channels pages of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

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This Item
I6138R9525SML1821
Efaroxan hydrochloride ≥98% (HPLC)

Sigma-Aldrich

E3263

Efaroxan hydrochloride

Idazoxan hydrochloride

Sigma-Aldrich

I6138

Idazoxan hydrochloride

RX 821002 hydrochloride solid, ≥98% (HPLC)

Sigma-Aldrich

R9525

RX 821002 hydrochloride

Imidafenacin hydrochloride ≥95% (HPLC)

Sigma-Aldrich

SML1821

Imidafenacin hydrochloride

assay

≥98% (HPLC)

assay

-

assay

≥98% (HPLC)

assay

≥95% (HPLC)

Quality Level

100

Quality Level

100

Quality Level

100

Quality Level

100

solubility

H2O: >20 mg/mL

solubility

H2O: 50 mg/mL

solubility

H2O: >20 mg/mL

solubility

H2O: 15 mg/mL, clear

Gene Information

human ... ADRA1A(148), ADRA1B(147), ADRA1D(146), ADRA2A(150), ADRA2B(151), ADRA2C(152)

Gene Information

human ... ADRA2A(150), ADRA2B(151), ADRA2C(152)

Gene Information

human ... ADRA2A(150), ADRA2B(151), ADRA2C(152)

Gene Information

-

pictograms

Skull and crossbones
GHS06

signalword

Danger

hcodes

H301

Hazard Classifications

Acute Tox. 3 Oral

Storage Class

6.1C - Combustible acute toxic Cat.3 / toxic compounds or compounds which causing chronic effects

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Faceshields, Gloves, type P2 (EN 143) respirator cartridges

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