R134

Rilmenidine hemifumarate salt

solid

• Sinónimos: N-(Dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine hemifumarate salt, Oxaminozoline hemifumarate salt, Rilmenidene hemifumarate salt
• Fórmula empírica (notación de Hill): C₁₀H₁₆N₂O · 0.5C₄H₄O₄
• Número CAS: 207572-68-7
• Peso molecular: 238.28
• NACRES: NA.77
• PubChem Substance ID: 24277752
• UNSPSC Code: 12352200
• MDL number: MFCD09878261
• Form: solid

Propiedades

• form: solid
• Quality Segment: 100
• color: white
• solubility: DMSO: >10 mg/mL, H₂O: insoluble
• originator: Servier
• SMILES string: OC(=O)\C=C\C(O)=O.C1CN=C(NC(C2CC2)C3CC3)O1.C4CN=C(NC(C5CC5)C6CC6)O4
• InChI: 1S/2C10H16N2O.C4H4O4/c2*1-2-7(1)9(8-3-4-8)12-10-11-5-6-13-10;5-3(6)1-2-4(7)8/h2*7-9H,1-6H2,(H,11,12);1-2H,(H,5,6)(H,7,8)/b;;2-1+
• InChI key: LZFATBMLSYHRTC-WXXKFALUSA-N
• Gene Information: human ... NISCH(11188)

Descripción

Biochem/physiol Actions

Selective I₁ imidazoline receptor agonist.

Features and Benefits

This compound is featured on the Imidazoline Binding Sites page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

This compound was developed by Servier. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Información de seguridad

• ¿Qué está pasando?: WGK 3
• Punto de inflamación (°F): Not applicable
• Punto de inflamación (°C): Not applicable
• EPI (equipos de protección individual): Eyeshields, Gloves, type N95 (US)
• Pictogramas: GHS06
• Palabra de advertencia: Danger
• Códigos de peligro: H301
• Indicaciones de precaución: P264 - P270 - P301 + P310 - P405 - P501
• Hazard Classifications: Acute Tox. 3 Oral
• Clase de almacenamiento: 6.1C - Combustible acute toxic Cat.3 / toxic compounds or compounds which causing chronic effects