M4603

Acetyl-[Nle⁴, Asp⁵, D-2-Nal⁷, Lys¹⁰]-cyclo-α-Melanocyte Stimulating Hormone Amide Fragment 4-10

≥95% (HPLC), Melanocortin-4 receptor antagonist

• Synonym(e): SHU9119
• Empirische Formel (Hill-System): C₅₄H₇₁N₁₅O₉
• Molekulargewicht: 1074.24
• UNSPSC Code: 51111800
• NACRES: NA.32
• MDL number: MFCD02093607

Eigenschaften

• Produktname: Acetyl-[Nle⁴, Asp⁵, D-2-Nal⁷, Lys¹⁰]-cyclo-α-Melanocyte Stimulating Hormone Amide Fragment 4-10, ≥95% (HPLC)
• Quality Segment: 200
• assay: ≥95% (HPLC)
• UniProt accession no.: P01189
• storage temp.: −20°C
• Gene Information: human ... POMC(5443)

Beschreibung

Biochem/physiol Actions

Screening analogs of the cyclic lactam melanocortin agonist MTII led to the identification of the agoutimimetic SHU9119. This compound shares pharmacological properties with the agouti peptide in that it is a potent antagonist of the melanocortin-4 receptor and a less potent antagonist of the melanocortin-3 receptor.

Sicherheitshinweise

• Lagerklasse: 11 - Combustible Solids
• wgk: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable
• ppe: Eyeshields, Gloves, type N95 (US)