P2959

PD 142,893

≥97% (HPLC)

• Synonym(e): N-Acetyl-β-Phenyl-D-Phe-Leu-Asp-Ile-Ile-Trp
• Empirische Formel (Hill-System): C₅₀H₆₅N₇O₁₀
• CAS-Nummer: 155893-16-6
• Molekulargewicht: 924.09
• UNSPSC Code: 12352200
• MDL number: MFCD00467201

Eigenschaften

• assay: ≥97% (HPLC)
• storage temp.: −20°C
• SMILES string: CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](NC(C)=O)C(c1ccccc1)c2ccccc2)[C@@H](C)CC)C(=O)N[C@@H](Cc3c[nH]c4ccccc34)C(O)=O

Beschreibung

General description

Contains the conserved endothelin sequence, His-Leu-Asp-Ile-Ile-Trp, with His replaced by a bulky aromatic moiety.

Biochem/physiol Actions

Non-selective endothelin receptor antagonist.

Sicherheitshinweise

• Lagerklasse: 13 - Non Combustible Solids
• wgk: WGK 3
• flash_point_f: Not applicable
• flash_point_c: Not applicable
• ppe: Eyeshields, Gloves, type N95 (US)