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5-BDBD

Name: 5-BDBD
Brand: SIGMA

≥98% (HPLC), P2X4 inhibitor, powder

Synonym(s):

5-(3-Bromophenyl)-1,3-dihydro-2H-Benzofuro[3,2-e]-1,4-diazepin-2-one

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About This Item

Empirical Formula (Hill Notation):

C₁₇H₁₁BrN₂O₂

CAS Number:

768404-03-1

Molecular Weight:

355.19

UNSPSC Code:

12352200

PubChem Substance ID:

329824730

NACRES:

NA.77

MDL number:

MFCD18086878

Assay:

≥98% (HPLC)

Form:

powder

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Properties

Product Name

5-BDBD, ≥98% (HPLC)

Quality Segment

100

assay

≥98% (HPLC)

form

powder

color

white to beige

solubility

DMSO: 15 mg/mL (clear solution)

storage temp.

2-8°C

SMILES string

Brc1cccc(c1)C2=NCC(=O)Nc3c2oc4ccccc34

InChI

1S/C17H11BrN2O2/c18-11-5-3-4-10(8-11)15-17-16(20-14(21)9-19-15)12-6-1-2-7-13(12)22-17/h1-8H,9H2,(H,20,21)

InChI key

NKYMVQPXXTZHSF-UHFFFAOYSA-N

Description

Biochem/physiol Actions

5-BDBD is a specific inhibitor of P2X4.

5-BDBD is a specific inhibitor of P2X4. The compound inhibits P2X4 currents in CHO cells with an IC₅₀ of 500 nM.

In native tissues, 5-BDBD is considered as a beneficial antagonist to analyze the effect of P2X receptors (P2XRs) subtype P2X4R.

Features and Benefits

This compound is featured on the P2 Receptors: P2X Ion Channel Family page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

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Show Differences

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This Item	SML0617	SML0775	D0444
Sigma-Aldrich SML0450 5-BDBD	Sigma-Aldrich SML0617 A-804598	Sigma-Aldrich SML0775 PZ-II-029	Sigma-Aldrich D0444 DT-2 trifluoroacetate salt
description ≥98% (HPLC)	description ≥98% (HPLC)	description ≥98% (HPLC)	description ≥95% (HPLC), film
assay ≥98% (HPLC)	assay ≥98% (HPLC)	assay ≥98% (HPLC)	assay ≥95% (HPLC)
form powder	form powder	form powder	form film
Quality Level 100	Quality Level 100	Quality Level 100	Quality Level 200
storage temp. 2-8°C	storage temp. 2-8°C	storage temp. 2-8°C	storage temp. −20°C
solubility DMSO: 15 mg/mL (clear solution)	solubility DMSO: 10 mg/mL, clear	solubility DMSO: 10 mg/mL, clear	solubility H₂O: 0.5 mg/mL, clear
color white to beige	color white to beige	color white to light brown	color colorless to white

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Storage Class

11 - Combustible Solids

WGK

WGK 3

Flash Point (°F)

Not applicable

Flash Point (°C)

Not applicable

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