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Merck

Surface charge switching nanoparticles for magnetic resonance imaging.

International journal of pharmaceutics (2014-05-27)
Dong Jin Lee, Young Taik Oh, Eun Seong Lee
ABSTRACT

In this study, polypeptide-based nanoparticles [constituted using poly(L-lysine) coupled with deoxycholic acid (DOCA) and conjugated with 2,3-dimethylmaleic acid (DMA)] have high tumor selectivity once electrostatically switched by the acidic milieu of solid tumors. These nanoparticles exhibited a significantly increased in vitro cellular uptake and high accumulation in the acidic tumor site in vivo. Consequently, Fe3O4-loaded nanoparticles enabled high contrast magnetic resonance (MR) imaging of the tumor in vivo.

MATERIALS
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Brand
Product Description

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Triethylamine, BioUltra, ≥99.5% (GC)
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Acetic acid, ≥99.5%, FCC, FG
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Acetic acid, natural, ≥99.5%, FG
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N,N-Dimethylformamide, anhydrous, 99.8%
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Lauric acid, ≥98%, FCC, FG
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Acetic acid-12C2, 99.9 atom % 12C
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Lauric acid, natural, ≥98%, FCC, FG
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Triethylamine, ≥99.5%
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Triethylamine, ≥99.5%
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Triethylamine, puriss. p.a., ≥99.5% (GC)
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Acetic acid solution, suitable for HPLC
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Diethyl ether, suitable for HPLC, ≥99.9%, inhibitor-free
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Acetic acid, glacial, puriss., meets analytical specification of Ph. Eur., BP, USP, FCC, 99.8-100.5%
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Diethyl ether, reagent grade, ≥98%, contains ≤2% ethanol and ≤10ppm BHT as inhibitor
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N,N-Dimethylformamide, ACS reagent, ≥99.8%
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