SML2032

Win6mer trifluoroacetate salt

≥98% (HPLC)

• Synonym(e): Ac-ARTEVY-NH2 trifluouroaceate salt
• Empirische Formel (Hill-System): C₃₄H₅₄N₁₀O₁₁ · xC₂HF₃O₂
• CAS-Nummer: 2222444-20-2
• Molekulargewicht: 778.85 (free base basis)
• UNSPSC-Code: 12352200
• NACRES: NA.77

Eigenschaften

• Assay: ≥98% (HPLC)
• Form: film (Clear)
• Farbe: white to off-white
• Versandbedingung: wet ice
• Lagertemp.: −20°C
• SMILES String: C[C@H](NC(C)=O)C(N[C@H](C(N[C@@](C(N[C@H](C(N[C@H](C(N[C@H](C(N)=O)CC1=CC=C(C=C1)O)=O)C(C)C)=O)CCC(O)=O)=O)([H])[C@H](O)C)=O)CCCNC(N)=N)=O

Beschreibung

Biochem./physiol. Wirkung

Win6mer is a potent and specific inhibitor of MLL1 and SETd1A histone H3 lysine 4 (H3K4) methyltransferase complexes that does not inhibit MLL2-4 or SETd1B complexes. Win6mer potently binds to WDR5 in a 310-helical conformation. It does not inhibit isolated SET domain activity.

Sicherheitshinweise

• Lagerklassenschlüssel: 11 - Combustible Solids
• WGK: WGK 3
• Flammpunkt (°F): Not applicable
• Flammpunkt (°C): Not applicable