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Targeted protein S-nitrosylation of ACE2 inhibits SARS-CoV-2 infection.

Nature chemical biology (2022-09-30)
Chang-Ki Oh, Tomohiro Nakamura, Nathan Beutler, Xu Zhang, Juan Piña-Crespo, Maria Talantova, Swagata Ghatak, Dorit Trudler, Lauren N Carnevale, Scott R McKercher, Malina A Bakowski, Jolene K Diedrich, Amanda J Roberts, Ashley K Woods, Victor Chi, Anil K Gupta, Mia A Rosenfeld, Fiona L Kearns, Lorenzo Casalino, Namir Shaabani, Hejun Liu, Ian A Wilson, Rommie E Amaro, Dennis R Burton, John R Yates, Cyrus Becker, Thomas F Rogers, Arnab K Chatterjee, Stuart A Lipton
ABSTRACT

Prevention of infection and propagation of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is a high priority in the Coronavirus Disease 2019 (COVID-19) pandemic. Here we describe S-nitrosylation of multiple proteins involved in SARS-CoV-2 infection, including angiotensin-converting enzyme 2 (ACE2), the receptor for viral entry. This reaction prevents binding of ACE2 to the SARS-CoV-2 spike protein, thereby inhibiting viral entry, infectivity and cytotoxicity. Aminoadamantane compounds also inhibit coronavirus ion channels formed by envelope (E) protein. Accordingly, we developed dual-mechanism aminoadamantane nitrate compounds that inhibit viral entry and, thus, the spread of infection by S-nitrosylating ACE2 via targeted delivery of the drug after E protein channel blockade. These non-toxic compounds are active in vitro and in vivo in the Syrian hamster COVID-19 model and, thus, provide a novel avenue to pursue therapy.

MATERIALS
Product Number
Brand
Product Description

Sigma-Aldrich
NitroSynapsin hydrochloride, ≥98% (HPLC)
Sigma-Aldrich
Fetal Bovine Serum, non-USA origin, sterile-filtered, suitable for cell culture