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  • One-pot primary aminomethylation of aryl and heteroaryl halides with sodium phthalimidomethyltrifluoroborate.

One-pot primary aminomethylation of aryl and heteroaryl halides with sodium phthalimidomethyltrifluoroborate.

Organic letters (2012-05-18)
Norio Murai, Masayuki Miyano, Masahiro Yonaga, Keigo Tanaka
PMID22591586
ABSTRACT

A one-pot primary aminomethylation of aryl halides, triflates, mesylates, and tosylates via Suzuki-Miyaura cross-coupling reactions with sodium phthalimidomethyltrifluoroborate followed by deamidation with ethylenediamine is reported.

MATERIALS
Product Number
Brand
Product Description
83000
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304506
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