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CHRM1

cholinergic receptor, muscarinic 1

Synonyms:
HM1, M1, M1R
Species:
UniProtKB ID:
Gene ID:
  • Human(1128) Summary: The muscarinic cholinergic receptors belong to a larger family of G protein-coupled receptors. The functional diversity of these receptors is defined by the binding of acetylcholine and includes cellular responses such as adenylate cyclase inhibition, phosphoinositide degeneration, and potassium channel mediation. Muscarinic receptors influence many effects of acetylcholine in the central and peripheral nervous system. The muscarinic cholinergic receptor 1 is involved in mediation of vagally-induced bronchoconstriction and in the acid secretion of the gastrointestinal tract. The gene encoding this receptor is localized to 11q13. [provided by RefSeq, Jul 2008]
  • Mouse(12669) cholinergic receptor, muscarinic 1, CNS
  • Rat(25229) cholinergic receptor, muscarinic 1
  • domestic guinea pig(100728041) cholinergic receptor, muscarinic 1
  • domestic cat(493664) cholinergic receptor, muscarinic 1
  • domestic cat(101093801) cholinergic receptor, muscarinic 1
  • dog(483776) cholinergic receptor, muscarinic 1
  • sheep(101117029) cholinergic receptor, muscarinic 1
  • cow(281684) cholinergic receptor, muscarinic 1
  • Horse(100064117) cholinergic receptor, muscarinic 1
  • naked mole-rat(101702102) cholinergic receptor, muscarinic 1

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Small Molecule - Agonist

Product Number
Description
Species
Pilocarpine hydrochloride, European Pharmacopoeia (EP) Reference Standard,
Species
human
Pilocarpine nitrate for system suitability, European Pharmacopoeia (EP) Reference Standard,
Species
human
Pilocarpine hydrochloride, phyproof® Reference Substance,
Species
human
Pilocarpine Hydrochloride, Pharmaceutical Secondary Standard; Certified Reference Material,
Species
human
Pilocarpine hydrochloride, United States Pharmacopeia (USP) Reference Standard,
Species
human

Small Molecule - Antagonist

Product Number
Description
Species
(−)-Scopolamine hydrochloride, analytical standard,
Species
human
Procyclidine hydrochloride, ,
Species
human
Benztropine mesylate, ≥98% (HPLC),
Species
human
Pirenzepine dihydrochloride, ≥98% (TLC), powder,
Species
human
Quinuclidine, 97%,
Species
rat

Antibodies

Product Number
Description
Species Reactivity
Application
Anti-Muscarinic Acetylcholine Receptor m1 Antibody, Chemicon®, from rabbit,
Species Reactivity
mouse, rat
Application
immunohistochemistry
western blot

Small Molecule - Inhibitor

Product Number
Description
Species
Harmaline, ≥95%,
Species
human, rat

Small Molecule - Ligand

Product Number
Description
Species
Aminobenztropine, solid,
Species
human

Proteins

Product Number
Description
Species
ChemiScreen Membrane Preparation Human Recombinant M1 Muscarinic Acetylcholine Receptor, Human M1 GPCR membrane prepation for Radioligand binding Assays.,
Species
human

esiRNA

Product Number
Description
Species
MISSION® esiRNA, targeting human CHRM1,
Species
human